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词汇
conophylline
释义
conophylline
是从小叶狗牙花中提取出来的新的长春碱类衍生物。在体外可使K-ras-NRK和K-ras-NIH细胞系出现正常表型,并使K-ras-NRK细胞对2-脱氧葡萄糖的摄取减少,但它对K-ras-NRK细胞系的抑制作用是可逆的,conophylline还可抑制移植的K-ras-NIH3T3和K-ras-NRK肿瘤在裸鼠体内的生长,对荷L1210白血病的裸鼠生长无影响。
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更新时间:2026/11/11 13:21:25